SCHEMBL20136097

SCHEMBL20136097

COC1CCC(c2nccnc2N)CC1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
TYK2 P29597 1/20 0.37
JAK3 P52333 1/20 0.37
MAP4K4 O95819 1/20 0.34
PARP1 P09874 1/20 0.33
RET P07949 1/20 0.32
PDE10A Q9Y233 2/20 0.31
PIK3CA P42336 1/20 0.31
GRM1 Q13255 1/20 0.31
BACE1 P56817 1/20 0.30
BTK Q06187 1/20 0.30
USP2 O75604 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
ALOX15 P16050 1/20 0.30
GFER P55789 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9900636 0.84 NEK2 (0.34) USP2GAAMAPTALOX15GFER
SCHEMBL30154873 0.84 NEK2 (0.34) USP2GAAMAPTALOX15GFER
SCHEMBL30536162 0.79 JAK2 (0.39) JAK2JAK1TYK2JAK3MAP4K4
SCHEMBL28563124 0.75 TDO2 (0.37) JAK2JAK1TYK2JAK3BACE1
SCHEMBL30536195 0.75 NOS3 (0.39) JAK2JAK1TYK2JAK3MAP4K4
SCHEMBL28076460 0.72 HRH4 (0.41) JAK2JAK1TYK2JAK3MAPT
SCHEMBL16053346 0.72 OPRL1 (0.40) PDE10A
SCHEMBL21300026 0.72 ALOX5AP (0.37) JAK2JAK1TYK2JAK3MAP4K4
SCHEMBL22089675 0.70 JAK2 (0.36) JAK2JAK1TYK2JAK3PARP1
SCHEMBL482014 0.69 MAPK1 (0.43) MAP4K4PARP1PIK3CAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063143-B1 AMINOHETEROARYL BENZAMIDES AS KINASE INHIBITORS NOVARTIS AG (CH) 2018-05-16 EP disclosed