SCHEMBL28563124

SCHEMBL28563124

Nc1nccnc1C1CCCCC1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 3/20 0.37
HRH2 P25021 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
CYP11B2 P19099 1/20 0.34
FFAR2 O15552 3/20 0.34
ADK P55263 1/20 0.33
BACE1 P56817 1/20 0.33
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
NISCH Q9Y2I1 1/20 0.32
TNK2 Q07912 2/20 0.32
FGFR2 P21802 1/20 0.32
DGAT1 O75907 1/20 0.32
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
TYK2 P29597 1/20 0.32
JAK3 P52333 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9900636 0.89 NEK2 (0.34) GAA
SCHEMBL30154873 0.89 NEK2 (0.34) GAA
SCHEMBL2355700 0.84 CYP11B2 (0.40) TDO2HRH2HRH3CYP11B2KDM4E
SCHEMBL16053346 0.79 OPRL1 (0.40) TNK2
SCHEMBL28076460 0.79 HRH4 (0.41) HRH3TNK2JAK2JAK1TYK2
SCHEMBL9900173 0.77 BTK (0.46) JAK2JAK1JAK3
SCHEMBL9900029 0.77 BTK (0.46) JAK2JAK1JAK3
SCHEMBL15740601 0.75 TDO2 (0.36) TDO2HRH2HRH3CYP11B2FFAR2
SCHEMBL20136097 0.75 JAK2 (0.37) BACE1GAAJAK2JAK1TYK2
SCHEMBL7937826 0.74 NISCH (0.36) TDO2CYP11B2FFAR2KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112142715-A 2-amino-5-heterocyclic group substituted pyrazine derivative and application thereof 鲁南制药集团股份有限公司 2020-12-29 CN disclosed