SCHEMBL20138980

SCHEMBL20138980

C=CC(=O)Nc1ccc(Nc2ncnc3[nH]c(-c4ccc(Oc5ccccc5)cc4)cc23)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.67
ERBB2 P04626 4/20 0.67
BTK Q06187 6/20 0.61
KCNH2 Q12809 1/20 0.59
FYN P06241 4/20 0.56
SRC P12931 4/20 0.56
VCP P55072 1/20 0.56
TGM2 P21980 1/20 0.55
RET P07949 1/20 0.51
TTBK1 Q5TCY1 1/20 0.48
TTBK2 Q6IQ55 1/20 0.48
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20139083 0.93 EGFR (0.70) EGFRERBB2BTKKCNH2FYN
SCHEMBL20139118 0.86 EGFR (0.64) EGFRERBB2BTKKCNH2FYN
SCHEMBL20139048 0.83 SRC (0.59) EGFRERBB2BTKKCNH2FYN
SCHEMBL7237980 0.80 EGFR (0.84) EGFRERBB2BTKKCNH2FYN
SCHEMBL7239977 0.80 EGFR (1.00) EGFRERBB2BTKFYNSRC
SCHEMBL690318 0.77 TGM2 (0.71) EGFRERBB2BTKKCNH2FYN
SCHEMBL20139002 0.77 PIK3CD (0.55) EGFRERBB2BTKKCNH2FYN
SCHEMBL20150686 0.77 EGFR (0.50) EGFRERBB2BTKKCNH2FYN
SCHEMBL7241722 0.76 EGFR (0.76) EGFRERBB2BTKKCNH2FYN
SCHEMBL7238977 0.76 EGFR (0.73) EGFRERBB2BTKKCNH2FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018088780-A1 NOVEL PYRROLOPYRIMIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2018-05-17 WO claimed
WO-2018088780-A1 NOVEL PYRROLOPYRIMIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2018-05-17 WO disclosed