SCHEMBL20139009

SCHEMBL20139009

C=CC(=O)Nc1cccc(Nc2ncnc3[nH]c(-c4ccc(C(=O)N5CCNCC5)cc4)cc23)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.54
SRC P12931 5/20 0.54
BTK Q06187 3/20 0.54
BLK P51451 2/20 0.54
ITK Q08881 1/20 0.54
MKNK2 Q9HBH9 3/20 0.49
RIPK1 Q13546 1/20 0.49
PIK3CD O00329 2/20 0.47
KCNH2 Q12809 1/20 0.45
ERBB2 P04626 3/20 0.45
FYN P06241 3/20 0.45
BMX P51813 1/20 0.45
JAK3 P52333 1/20 0.45
ERBB4 Q15303 1/20 0.45
BRAF P15056 1/20 0.44
TNNI3K Q59H18 1/20 0.44
VCP P55072 1/20 0.44
CCNC P24863 1/20 0.44
CDK8 P49336 1/20 0.44
CSF1R P07333 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20150991 0.91 EGFR (0.53) EGFRSRCBTKBLKITK
SCHEMBL20139048 0.83 SRC (0.59) EGFRSRCBTKBLKPIK3CD
SCHEMBL20139429 0.82 JAK1 (0.59) EGFRBTKERBB2JAK3CSF1R
SCHEMBL29538618 0.82 JAK1 (0.59) EGFRBTKERBB2JAK3CSF1R
SCHEMBL21484334 0.81 ERBB2 (0.62) EGFRSRCERBB2JAK3
Methylpiperazine SCHEMBL4771183 0.80 RIPK1 (0.49) BTKMKNK2RIPK1BRAFTNNI3K
SCHEMBL20139083 0.79 EGFR (0.70) EGFRSRCBTKPIK3CDKCNH2
SCHEMBL20138988 0.79 EGFR (0.60) EGFRBTKPIK3CDERBB2JAK3
SCHEMBL20139788 0.79 PIK3CD (0.49) EGFRSRCBTKBLKPIK3CD
SCHEMBL20150686 0.79 EGFR (0.50) EGFRSRCBTKBLKITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018088780-A1 NOVEL PYRROLOPYRIMIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2018-05-17 WO claimed
WO-2018088780-A1 NOVEL PYRROLOPYRIMIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2018-05-17 WO disclosed