SCHEMBL20139669

SCHEMBL20139669

O=C/C=C(\c1ccccc1)c1ccc(Br)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 1/20 0.44
AKR1C3 P42330 1/20 0.43
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
TP53 P04637 1/20 0.42
HPGD P15428 1/20 0.42
ALDH1A1 P00352 5/20 0.41
MAPT P10636 4/20 0.41
TDP1 Q9NUW8 3/20 0.41
ALOX12 P18054 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GAA P10253 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 1/20 0.40
NFKB1 P19838 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1320539 1.00 CYP1B1 (0.44) CYP1B1AKR1C3MEN1KMT2ANPC1
SCHEMBL6387039 0.92 CES2 (0.48) CYP1B1MEN1KMT2ARAB9AHPGD
SCHEMBL376723 0.87 ALDH1A1 (0.48) MEN1KMT2AHPGDALDH1A1MAPT
SCHEMBL11285264 0.81 CYP3A4 (0.58) MEN1KMT2ANPC1RAB9AHPGD
SCHEMBL11285263 0.81 CYP3A4 (0.58) MEN1KMT2ANPC1RAB9AHPGD
SCHEMBL11288939 0.81 CYP3A4 (0.58) MEN1KMT2ANPC1RAB9AHPGD
SCHEMBL29016164 0.80 CES2 (0.55) CYP1B1ALDH1A1MAPTCES2CES1
SCHEMBL18885235 0.80 CES2 (0.55) CYP1B1AKR1C3MEN1KMT2ANPC1
SCHEMBL10579805 0.80 CES2 (0.55) CYP1B1ALDH1A1MAPTCES2CES1
SCHEMBL9472917 0.79 SMN1; SMN2 (0.48) MEN1KMT2ANPC1RAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538522-A1 ROR GAMMA MODULATORS Bristol-Myers Squibb Company (US) 2019-09-18 EP disclosed
WO-2018089406-A1 ROR GAMMA MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed