SCHEMBL20139744

SCHEMBL20139744

C[C@H]1CN(c2cccc3cc[nH]c23)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.46
HDAC1 Q13547 1/20 0.42
GPR119 Q8TDV5 2/20 0.42
SUV39H2 Q9H5I1 2/20 0.41
NR1H2 P55055 8/20 0.40
IDO1 P14902 1/20 0.40
NR1H3 Q13133 7/20 0.39
SETD7 Q8WTS6 1/20 0.39
MAPT P10636 1/20 0.37
BCHE P06276 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20141652 0.83 HDAC1 (0.47) MAP4K4HDAC1GPR119SUV39H2NR1H2
SCHEMBL20141654 0.83 HDAC1 (0.47) MAP4K4HDAC1GPR119SUV39H2NR1H2
SCHEMBL5205461 0.83 IDO1 (0.48) GPR119IDO1MAPTBCHE
SCHEMBL30885785 0.83 IDO1 (0.48) GPR119IDO1MAPTBCHE
SCHEMBL28520979 0.82 MAP4K4 (0.49) MAP4K4HDAC1GPR119SUV39H2NR1H2
SCHEMBL23602022 0.79 MAP4K4 (0.53) MAP4K4HDAC1GPR119SUV39H2NR1H2
SCHEMBL13999776 0.78 HDAC1 (0.49) MAP4K4HDAC1GPR119NR1H2NR1H3
SCHEMBL13384125 0.78 HDAC1 (0.54) MAP4K4HDAC1GPR119SUV39H2NR1H2
SCHEMBL28600264 0.78 DRD2 (0.50) MAP4K4HDAC1GPR119SUV39H2
SCHEMBL29799403 0.78 DRD2 (0.50) MAP4K4HDAC1GPR119SUV39H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed