SCHEMBL20141652

SCHEMBL20141652

CC1CN(c2cccc3cn[nH]c23)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.47
MAP4K4 O95819 1/20 0.47
GPR119 Q8TDV5 2/20 0.45
HTR1A P08908 1/20 0.43
ACACB O00763 2/20 0.42
SUV39H2 Q9H5I1 2/20 0.40
UCHL1 P09936 1/20 0.39
NR1H2 P55055 5/20 0.39
IDO1 P14902 1/20 0.38
NR1H3 Q13133 4/20 0.38
SPR P35270 2/20 0.38
SETD7 Q8WTS6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20141654 1.00 HDAC1 (0.47) HDAC1MAP4K4GPR119HTR1AACACB
SCHEMBL20139744 0.83 MAP4K4 (0.46) HDAC1MAP4K4GPR119SUV39H2NR1H2
SCHEMBL28520979 0.81 MAP4K4 (0.49) HDAC1MAP4K4GPR119SUV39H2NR1H2
SCHEMBL17114986 0.80 MAP4K4 (0.47) HDAC1MAP4K4GPR119SUV39H2NR1H2
SCHEMBL17114988 0.80 MAP4K4 (0.47) HDAC1MAP4K4GPR119SUV39H2NR1H2
SCHEMBL23602022 0.79 MAP4K4 (0.53) HDAC1MAP4K4GPR119HTR1ASUV39H2
SCHEMBL20831929 0.77 TRPC5 (0.46) HDAC1MAP4K4GPR119SUV39H2IDO1
SCHEMBL13999776 0.77 HDAC1 (0.49) HDAC1MAP4K4GPR119NR1H2NR1H3
SCHEMBL29799403 0.76 DRD2 (0.50) HDAC1MAP4K4GPR119SUV39H2
SCHEMBL24719091 0.76 DRD2 (0.50) HDAC1MAP4K4GPR119SUV39H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed