SCHEMBL20140039

SCHEMBL20140039

COC(=O)c1c(-c2ccccc2)cnn1CCNC(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 2/20 0.44
SKP1 P63208 2/20 0.44
SKP2 Q13309 2/20 0.44
DRD2 P14416 5/20 0.43
SMN1; SMN2 Q16637 1/20 0.40
MALT1 Q9UDY8 1/20 0.39
IDO1 P14902 1/20 0.39
PDCD1 Q15116 1/20 0.39
CD274 Q9NZQ7 1/20 0.39
ITGA4 P13612 1/20 0.39
ITGB7 P26010 1/20 0.39
PTGIR P43119 2/20 0.39
AKT1 P31749 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA3 P34903 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20140432 0.84 CKS1B (0.45) CKS1BSKP1SKP2DRD2SMN1; SMN2
SCHEMBL20140105 0.83 CKS1B (0.44) CKS1BSKP1SKP2DRD2SMN1; SMN2
SCHEMBL20139538 0.81 DRD2 (0.40) DRD2
SCHEMBL20401167 0.80 DRD2 (0.39) DRD2
SCHEMBL29544458 0.78 GAA (0.40) DRD2SMN1; SMN2
SCHEMBL1314087 0.76 SMN1; SMN2 (0.47) CKS1BSKP1SKP2DRD2SMN1; SMN2
SCHEMBL2552113 0.76 BCHE (0.47) DRD2
SCHEMBL18187542 0.74 IDO1 (0.43) DRD2SMN1; SMN2IDO1AKT1SIGMAR1
SCHEMBL1313637 0.73 BRD9 (0.46) CKS1BSKP1SKP2DRD2IDO1
SCHEMBL20027667 0.73 LPAR1 (0.49) PTGIRGABRA1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed