SCHEMBL20140105

SCHEMBL20140105

CC(C)(C)OC(=O)NCCn1ncc(-c2ccccc2)c1CCl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 1/20 0.44
SKP1 P63208 1/20 0.44
SKP2 Q13309 1/20 0.44
PTGIR P43119 2/20 0.42
DRD2 P14416 3/20 0.42
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CYP3A4 P08684 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
NCOA1 Q15788 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20140432 0.92 CKS1B (0.45) CKS1BSKP1SKP2PTGIRDRD2
SCHEMBL20140039 0.83 CKS1B (0.44) CKS1BSKP1SKP2PTGIRDRD2
SCHEMBL30239588 0.77 CYP3A4 (0.47) CKS1BSKP1SKP2DRD2SIGMAR1
SCHEMBL24931121 0.75 ALDH1A1 (0.45) HDAC3HDAC1HDAC8HDAC6SIGMAR1
SCHEMBL1313637 0.74 BRD9 (0.46) CKS1BSKP1SKP2DRD2SIGMAR1
SCHEMBL20140446 0.74 PTGIR (0.44) PTGIRSMN1; SMN2MEN1LMNAHTT
SCHEMBL28256776 0.72 NQO2 (0.54) CKS1BSKP1SKP2DRD2HDAC3
SCHEMBL17619511 0.72 ALDH1A1 (0.56) CKS1BSKP1SKP2DRD2SMN1; SMN2
SCHEMBL1949387 0.71 CKS1B (0.47) CKS1BSKP1SKP2DRD2SIGMAR1
SCHEMBL15936752 0.71 PDK2 (0.46) CKS1BSKP1SKP2DRD2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed