SCHEMBL20140432

SCHEMBL20140432

CC(C)(C)OC(=O)NCCn1ncc(-c2ccccc2)c1CO

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 2/20 0.45
SKP1 P63208 2/20 0.45
SKP2 Q13309 2/20 0.45
DRD2 P14416 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.41
MALT1 Q9UDY8 1/20 0.41
IDO1 P14902 1/20 0.41
PTGIR P43119 2/20 0.40
PDCD1 Q15116 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
SIGMAR1 Q99720 2/20 0.40
AKT1 P31749 1/20 0.40
BCHE P06276 1/20 0.39
SCN9A Q15858 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20140105 0.92 CKS1B (0.44) CKS1BSKP1SKP2DRD2SMN1; SMN2
SCHEMBL20140039 0.84 CKS1B (0.44) CKS1BSKP1SKP2DRD2SMN1; SMN2
SCHEMBL30239588 0.78 CYP3A4 (0.47) CKS1BSKP1SKP2DRD2IDO1
SCHEMBL1313637 0.77 BRD9 (0.46) CKS1BSKP1SKP2DRD2IDO1
SCHEMBL24931121 0.74 ALDH1A1 (0.45) SMN1; SMN2IDO1HDAC3HDAC1HDAC8
SCHEMBL28256776 0.73 NQO2 (0.54) CKS1BSKP1SKP2DRD2SMN1; SMN2
SCHEMBL17619511 0.73 ALDH1A1 (0.56) CKS1BSKP1SKP2DRD2SMN1; SMN2
SCHEMBL1949387 0.72 CKS1B (0.47) CKS1BSKP1SKP2DRD2IDO1
SCHEMBL20141217 0.72 CKS1B (0.42) CKS1BSKP1SKP2DRD2IDO1
SCHEMBL24376372 0.72 BRD4 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed