SCHEMBL20140127

SCHEMBL20140127

N#Cc1ccccc1N1CCCNCC1

nearest known ligand 0.87

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 3/20 0.51
AR P10275 1/20 0.49
DPP4 P27487 1/20 0.48
HTR6 P50406 4/20 0.48
HTR1A P08908 3/20 0.48
HTR7 P34969 3/20 0.48
HTR3A P46098 3/20 0.48
HTR2B P41595 1/20 0.48
HTR2A P28223 2/20 0.47
HTR5A P47898 2/20 0.47
HTR3E A5X5Y0 2/20 0.47
HTR3B O95264 2/20 0.47
HTR3D Q70Z44 2/20 0.47
HTR3C Q8WXA8 2/20 0.47
SIGMAR1 Q99720 2/20 0.47
NCF1 P14598 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
TSHR P16473 1/20 0.47
NFKB1 P19838 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL233169 0.93 ADRB1 (0.58) ADRB1HTR6HTR1AHTR7HTR3A
Hydrochloric Acid SCHEMBL29882725 0.91 ADRB1 (0.56) ADRB1HTR6HTR1AHTR7HTR3A
Hydrochloric Acid SCHEMBL20139829 0.91 ADRB1 (0.56) ADRB1HTR6HTR1AHTR7HTR3A
SCHEMBL829177 0.84 AR (0.65) ARHTR1AALDH1A1DRD2KDM4E
SCHEMBL30406641 0.84 AR (0.59) ARHTR1AALDH1A1DRD2DRD3
SCHEMBL6718397 0.83 DRD2 (0.53) ADRB1HTR6HTR1AHTR7HTR3A
SCHEMBL7524105 0.82 AR (0.62) ARHTR1AALDH1A1DRD2KDM4E
SCHEMBL31388194 0.82 AR (0.62) ARHTR1AALDH1A1DRD2KDM4E
SCHEMBL7528396 0.82 AR (0.62) ARHTR1AALDH1A1DRD2KDM4E
SCHEMBL1660394 0.82 AR (0.62) ARHTR1AALDH1A1DRD2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023186065-A1 A CYCLIN-DEPENDENT KINASE INHIBITOR Taizhou Eoc Pharma Co., Ltd. (CN) 2023-10-05 WO disclosed
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed
WO-2019238067-A1 PYRROLO [2, 3-B] PYRIDINES OR PYRROLO [2, 3-B] PYRAZINES AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2019-12-19 WO disclosed
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed