SCHEMBL6718397

SCHEMBL6718397

N#Cc1ccc(N2CCNCC2)cc1.N#Cc1ccccc1N1CCNCC1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.53
DRD3 P35462 1/20 0.53
ADRB1 P08588 5/20 0.51
HTR3E A5X5Y0 2/20 0.51
HTR3B O95264 2/20 0.51
HTR3A P46098 2/20 0.51
HTR3D Q70Z44 2/20 0.51
HTR3C Q8WXA8 2/20 0.51
SIGMAR1 Q99720 2/20 0.51
KDM4E B2RXH2 1/20 0.49
TP53 P04637 1/20 0.49
LTA4H P09960 1/20 0.46
OPRD1 P41143 1/20 0.46
CHRNA10 Q9GZZ6 1/20 0.46
CHRNA9 Q9UGM1 1/20 0.46
HTR6 P50406 2/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TSHR P16473 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL233169 0.89 ADRB1 (0.58) DRD2DRD3ADRB1HTR3EHTR3B
Hydrochloric Acid SCHEMBL20139829 0.87 ADRB1 (0.56) DRD2DRD3ADRB1HTR3EHTR3B
Hydrochloric Acid SCHEMBL29882725 0.87 ADRB1 (0.56) DRD2DRD3ADRB1HTR3EHTR3B
SCHEMBL6956744 0.85 KDM4E (0.63) DRD2DRD3ADRB1HTR3EHTR3B
SCHEMBL231077 0.85 KDM4E (0.63) DRD2DRD3ADRB1HTR3EHTR3B
Hydrochloric Acid SCHEMBL23303443 0.84 KDM4E (0.61) DRD2DRD3ADRB1HTR3EHTR3B
Hydrochloric Acid SCHEMBL376202 0.84 KDM4E (0.61) DRD2DRD3ADRB1HTR3EHTR3B
SCHEMBL20140127 0.83 ADRB1 (0.51) DRD2DRD3ADRB1HTR3EHTR3B
SCHEMBL24989037 0.80 KDM4E (0.58) DRD2DRD3ADRB1HTR3EHTR3B
SCHEMBL4228201 0.79 KDM4E (0.56) DRD2DRD3ADRB1HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313477-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2004-03-03 EP disclosed
US-20040038982-A1 Compounds and methods SMITHKLINE BEECHAM CORPORATION 2004-02-26 US disclosed
EP-1313477-A1 COMPOUNDS AND METHODS SmithKline Beecham Corporation (US) 2003-05-28 EP disclosed
WO-2002005819-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2002-01-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040038982-A1 Compounds and methods CCR5, CXCR3, CCR2 DRD2 645/4885DRD3 519/4885ADRB1 75/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.