SCHEMBL20140426

SCHEMBL20140426

Fc1c(-c2ccccc2)ccc(N2CCCC2)c1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.43
HTR7 P34969 2/20 0.43
HTR1A P08908 1/20 0.43
HTR2A P28223 1/20 0.43
HTR5A P47898 1/20 0.43
ALDH1A1 P00352 4/20 0.41
L3MBTL1 Q9Y468 4/20 0.41
KDM4E B2RXH2 3/20 0.41
TDP1 Q9NUW8 1/20 0.41
MAPT P10636 1/20 0.41
KEAP1 Q14145 1/20 0.40
PTGS2 P35354 1/20 0.40
HSD17B10 Q99714 2/20 0.39
AR P10275 1/20 0.39
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39
TP53 P04637 1/20 0.39
ALOX15 P16050 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAPK1 P28482 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10533047 0.77 ALOX5AP (0.53) ALDH1A1MAPTPTGS2HSD17B10ALOX5AP
SCHEMBL5352962 0.76 HTR7 (0.69) HTR6HTR7HTR1AHTR2AHTR5A
SCHEMBL27876080 0.75 HTR7 (0.67) HTR6HTR7HTR1AHTR2AHTR5A
SCHEMBL13039956 0.75 HTR7 (0.67) HTR6HTR7HTR1AHTR2AHTR5A
Hydrochloric Acid SCHEMBL27892728 0.73 HTR7 (0.65) HTR6HTR7HTR1AHTR2AHTR5A
SCHEMBL31402471 0.73 ALDH1A1 (0.36) ALDH1A1L3MBTL1KDM4EMAPTKEAP1
SCHEMBL4914927 0.73 HTR7 (0.73) HTR6HTR7HTR1AHTR2AHTR5A
SCHEMBL28618211 0.73 KDM4E (0.41) ALDH1A1L3MBTL1KDM4ETDP1MAPT
SCHEMBL19308566 0.73 ALDH1A1 (0.50) ALDH1A1L3MBTL1TDP1MAPTHSD17B10
Hydrochloric Acid SCHEMBL6570766 0.71 ALDH1A1 (0.57) HTR6HTR7HTR1AHTR2AHTR5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538522-A1 ROR GAMMA MODULATORS Bristol-Myers Squibb Company (US) 2019-09-18 EP disclosed
WO-2018089406-A1 ROR GAMMA MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed