SCHEMBL20140485

SCHEMBL20140485

COc1ccc(C(CC(=O)O)NC(=O)C2CC(CCO)C2)cn1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.51
ITGA4 P13612 1/20 0.51
CHRNA7 P36544 5/20 0.45
ITGB3 P05106 4/20 0.43
ITGA2B P08514 4/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
LMNA P02545 1/20 0.39
ACACB O00763 1/20 0.39
KCNK3 O14649 3/20 0.38
POLB P06746 1/20 0.38
P2RX3 P56373 2/20 0.38
P2RX2 Q9UBL9 2/20 0.38
CTSA P10619 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20140452 0.87 ITGB1 (0.53) ITGB1ITGA4CHRNA7ITGB3ITGA2B
SCHEMBL20158050 0.79 ITGB3 (0.62) ITGB1ITGB3ITGA2B
SCHEMBL20140803 0.79 ITGB3 (0.62) ITGB1ITGB3ITGA2B
SCHEMBL20142840 0.79 ITGB1 (0.43) ITGB1ITGA4CHRNA7ITGB3ITGA2B
SCHEMBL20142834 0.79 ITGB1 (0.43) ITGB1ITGA4CHRNA7ITGB3ITGA2B
SCHEMBL20140807 0.79 ITGB3 (0.62) ITGB1ITGB3ITGA2B
SCHEMBL29701366 0.79 ITGB3 (0.62) ITGB1ITGB3ITGA2B
SCHEMBL29701370 0.79 ITGB1 (0.43) ITGB1ITGA4CHRNA7ITGB3ITGA2B
SCHEMBL21317545 0.79 ITGB3 (0.62) ITGB1ITGB3ITGA2B
SCHEMBL20140536 0.79 ITGB1 (0.51) ITGB1ITGA4CHRNA7ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538526-A1 CYCLOBUTANE- AND AZETIDINE-CONTAINING MONO AND SPIROCYCLIC COMPOUNDS AS ALPHA V INTEGRIN INHIBITORS Bristol-Myers Squibb Company (US) 2019-09-18 EP disclosed
WO-2018089355-A1 CYCLOBUTANE- AND AZETIDINE-CONTAINING MONO AND SPIROCYCLIC COMPOUNDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed