SCHEMBL20141060

SCHEMBL20141060

C[C@H]1CN(c2cccc(N)c2)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 11/20 0.55
NR1H3 Q13133 10/20 0.54
MAP4K4 O95819 1/20 0.53
FAAH O00519 5/20 0.51
HDAC1 Q13547 1/20 0.50
SUV39H2 Q9H5I1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20139232 0.88 NR1H2 (0.55) NR1H2NR1H3FAAHSUV39H2
SCHEMBL30208177 0.88 NR1H2 (0.55) NR1H2NR1H3FAAHSUV39H2
SCHEMBL16580717 0.86 MAP4K4 (0.55) NR1H2NR1H3MAP4K4FAAHHDAC1
SCHEMBL17958723 0.86 MAP4K4 (0.55) NR1H2NR1H3MAP4K4FAAHHDAC1
SCHEMBL5465391 0.86 MAP4K4 (0.55) NR1H2NR1H3MAP4K4FAAHHDAC1
SCHEMBL20139199 0.86 FAAH (0.56) NR1H2NR1H3MAP4K4FAAHHDAC1
SCHEMBL15819221 0.86 FAAH (0.56) NR1H2NR1H3MAP4K4FAAHHDAC1
SCHEMBL16933542 0.86 NR1H2 (0.57) NR1H2NR1H3MAP4K4FAAHHDAC1
SCHEMBL20159043 0.84 CHRM2 (0.53) NR1H2NR1H3MAP4K4FAAHSUV39H2
SCHEMBL5782035 0.84 GPR119 (0.46) NR1H2NR1H3MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed