SCHEMBL20159043

SCHEMBL20159043

C[C@H]1CN(c2cccc(C#N)c2)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.53
CHRM1 P11229 1/20 0.53
NR1H2 P55055 12/20 0.52
NOTUM Q6P988 1/20 0.51
NR1H3 Q13133 11/20 0.51
FAAH O00519 3/20 0.48
SUV39H2 Q9H5I1 1/20 0.45
MAP4K4 O95819 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL705715 0.86 AR (0.53) NR1H2NR1H3SUV39H2MAP4K4
SCHEMBL705714 0.86 AR (0.53) NR1H2NR1H3SUV39H2MAP4K4
SCHEMBL30208177 0.84 NR1H2 (0.55) NR1H2NR1H3FAAHSUV39H2
SCHEMBL20139232 0.84 NR1H2 (0.55) NR1H2NR1H3FAAHSUV39H2
SCHEMBL20141060 0.84 NR1H2 (0.55) NR1H2NR1H3FAAHSUV39H2MAP4K4
SCHEMBL15819221 0.82 FAAH (0.56) NR1H2NR1H3FAAHMAP4K4
SCHEMBL20139199 0.82 FAAH (0.56) NR1H2NR1H3FAAHMAP4K4
SCHEMBL16933542 0.82 NR1H2 (0.57) NR1H2NR1H3FAAHSUV39H2MAP4K4
SCHEMBL688078 0.82 GPR119 (0.56) NOTUMFAAH
SCHEMBL29767485 0.81 CHRM4 (0.53) CHRM2MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed