SCHEMBL20141383

SCHEMBL20141383

CC(C)(C)OC(=O)NCCc1ccc(C#N)c(F)c1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.52
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CACNA1H O95180 5/20 0.44
EGLN2 Q96KS0 1/20 0.44
NAMPT P43490 1/20 0.43
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
NQO2 P16083 1/20 0.41
DAO P14920 1/20 0.41
AAK1 Q2M2I8 1/20 0.41
MAPT P10636 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27549593 0.89 TRPA1 (0.47) TRPA1CA1CA2CACNA1HEGLN2
SCHEMBL30751832 0.88 CTSS (0.47) TRPA1EGLN2CTSSCTSKNQO2
SCHEMBL21266053 0.88 CTSS (0.47) TRPA1EGLN2CTSSCTSKNQO2
SCHEMBL6928939 0.88 TRPA1 (0.54) TRPA1CACNA1HEGLN2NAMPTCTSS
SCHEMBL13171671 0.86 NSD2 (0.46) TRPA1CA1CA2CACNA1HNAMPT
SCHEMBL31432911 0.85 CA1 (0.48) CA1CA2CACNA1HAAK1MAPT
SCHEMBL7933824 0.84 TRPA1 (0.46) TRPA1CACNA1HEGLN2CTSSCTSK
SCHEMBL31432797 0.84 CA1 (0.47) CA1CA2CACNA1HMAPT
SCHEMBL16822026 0.84 KCNJ1 (0.43) TRPA1CA1CA2NAMPTCTSS
SCHEMBL5106289 0.84 CA1 (0.41) TRPA1CA1CA2NAMPTCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed