SCHEMBL7933824

SCHEMBL7933824

CC(C)(C)OC(=O)NCCc1cnc(Cc2ccc(C#N)c(F)c2)[nH]1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.46
CACNA1H O95180 8/20 0.41
EGLN2 Q96KS0 1/20 0.41
BCHE P06276 1/20 0.39
AAK1 Q2M2I8 3/20 0.39
NSD2 O96028 1/20 0.39
DAO P14920 1/20 0.39
PARP1 P09874 1/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
MAPT P10636 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20141383 0.84 TRPA1 (0.52) TRPA1CACNA1HEGLN2AAK1DAO
SCHEMBL7673651 0.80 CACNA1H (0.45) TRPA1CACNA1HEGLN2MAPTTDP1
SCHEMBL6928939 0.78 TRPA1 (0.54) TRPA1CACNA1HEGLN2NSD2CTSS
SCHEMBL6432281 0.78 DAO (0.42) CACNA1HDAO
Bromide SCHEMBL6409244 0.77 DAO (0.42) CACNA1HDAO
SCHEMBL27549593 0.77 TRPA1 (0.47) TRPA1CACNA1HEGLN2CTSSCTSK
SCHEMBL7183733 0.77 CYP11B1 (0.46) TRPA1CACNA1HEGLN2
SCHEMBL6433917 0.77 DAO (0.46) CACNA1HDAO
SCHEMBL28963038 0.76 CA12 (0.43) TRPA1CACNA1HEGLN2CTSSCTSK
SCHEMBL7743907 0.75 DAO (0.47) NSD2DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001017992-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed