SCHEMBL20141457

SCHEMBL20141457

CC(C)(C)[Si](C)(C)OC[C@@H]1CNCCN1c1ccc(F)cn1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
HDAC1 Q13547 1/20 0.36
HTR2C P28335 2/20 0.35
CHRNA7 P36544 2/20 0.35
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
KCNH2 Q12809 1/20 0.34
FPR2 P25090 1/20 0.34
SCN9A Q15858 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2B P41595 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31045993 0.84 CYP2D6 (0.50) CYP2D6SLC6A2SLC6A4SLC6A3HTR2C
SCHEMBL20133585 0.82 PLD1 (0.41) CYP2D6SLC6A2SLC6A4SLC6A3HTR2C
SCHEMBL20141404 0.78 FPR2 (0.48) SLC6A2SLC6A4SLC6A3HDAC8HDAC6
SCHEMBL20140978 0.77 MTOR (0.39) HDAC8HDAC6
SCHEMBL20133720 0.76 SLC6A2 (0.40) CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL20141556 0.76 SLC6A2 (0.40) CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL21360351 0.75 HDAC8 (0.44) HDAC8HDAC6
SCHEMBL15858056 0.73 HTR2C (0.45) HDAC8HDAC6HDAC1HTR2CKCNH2
SCHEMBL20142005 0.72 PLD1 (0.39) CYP2D6SLC6A2SLC6A4SLC6A3HTR2C
SCHEMBL30132155 0.71 CYP2D6 (0.35) CYP2D6SLC6A2SLC6A4SLC6A3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538091-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF Navitor Pharmaceuticals, Inc. (US) 2019-09-18 EP disclosed
WO-2018089499-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed