SCHEMBL20141712

SCHEMBL20141712

C[C@H]1CN(c2cccc3c(OC(=O)C(F)(F)F)c[nH]c23)CCN1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.39
BRPF1 P55201 2/20 0.36
BRD4 O60885 1/20 0.36
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 3/20 0.35
HPGD P15428 2/20 0.35
HSD17B10 Q99714 2/20 0.35
PMP22 Q01453 1/20 0.35
LMNA P02545 1/20 0.33
PRKCQ Q04759 3/20 0.33
HTR6 P50406 2/20 0.32
CDK1 P06493 1/20 0.32
CDK2 P24941 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
BIRC2 Q13490 2/20 0.32
XIAP P98170 1/20 0.32
PRKCD Q05655 1/20 0.32
PIM1 P11309 1/20 0.32
MCHR1 Q99705 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20139839 0.78 MAPT (0.38) HTR2CKDM4EALDH1A1HPGDHSD17B10
Trifluoroacetic Acid SCHEMBL20141711 0.72 HTR2C (0.39) HTR2CBRPF1BRD4ALDH1A1LMNA
SCHEMBL28172901 0.69 KDM4E (0.50) BRPF1BRD4KDM4EALDH1A1HPGD
SCHEMBL4590419 0.68 PDPK1 (0.40) BRPF1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL20142186 0.66 HTR6 (0.36) ALDH1A1HTR6
SCHEMBL23744700 0.66 HTR2C (0.59) HTR2CALDH1A1LMNA
SCHEMBL3219375 0.66 HTR2C (0.59) HTR2CALDH1A1LMNA
SCHEMBL3219365 0.66 HTR2C (0.59) HTR2CALDH1A1LMNA
SCHEMBL4244446 0.66 HTR6 (0.61) HTR2CKDM4EALDH1A1HPGDHSD17B10
SCHEMBL30345613 0.66 HTR2C (0.59) HTR2CALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed