SCHEMBL20142391

SCHEMBL20142391

CN(C)c1nc(Nc2ccc(C(F)(F)F)cc2)sc1C(=O)c1ccc(C(=O)O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
ADORA2A P29274 1/20 0.48
ADORA1 P30542 1/20 0.48
DHODH Q02127 1/20 0.47
MAPT P10636 4/20 0.47
SRD5A2 P31213 1/20 0.47
NPC1 O15118 6/20 0.47
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
RAB9A P51151 4/20 0.47
ALDH1A1 P00352 1/20 0.46
POLB P06746 1/20 0.46
CCNA2 P20248 5/20 0.45
CDK2 P24941 5/20 0.45
CFTR P13569 1/20 0.44
CDK5 Q00535 4/20 0.43
CDK5R1 Q15078 4/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20142501 0.90 CDK5 (0.49) ADORA3ADORA2AADORA1DHODHMAPT
SCHEMBL20142452 0.86 NPC1 (0.50) EPHX2ADORA3ADORA2AADORA1DHODH
SCHEMBL20142502 0.84 MEN1 (0.64) ADORA3ADORA2AADORA1DHODHMAPT
SCHEMBL20142497 0.83 CCNA2 (0.55) ADORA3ADORA2AADORA1DHODHMAPT
SCHEMBL20141966 0.83 MAPT (0.66) MAPTNPC1MEN1KMT2ARAB9A
SCHEMBL20142504 0.80 CCNA2 (0.49) ADORA3ADORA2AADORA1DHODHMAPT
SCHEMBL20142105 0.80 CDK5 (0.67) MAPTNPC1MEN1KMT2ARAB9A
SCHEMBL20142841 0.78 MAPT (0.63) ADORA3ADORA2AADORA1MAPTNPC1
SCHEMBL20142465 0.78 CDK5 (0.52) ADORA3ADORA2AADORA1DHODHMAPT
SCHEMBL20142402 0.78 NPC1 (0.57) DHODHMAPTNPC1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089902-A1 DIAMINOTHIAZOLE COMPOUNDS, COMPOSITIONS AND METHODS OF USE APOGEE BIOTECHNOLOGY CORPORATION (US) 2018-05-17 WO disclosed