SCHEMBL20142452

SCHEMBL20142452

CN(C)c1nc(Nc2ccc(OC(F)(F)F)cc2)sc1C(=O)c1ccc(C(=O)O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.50
MEN1 O00255 5/20 0.50
KMT2A Q03164 5/20 0.50
CDK5 Q00535 3/20 0.47
CDK5R1 Q15078 3/20 0.47
MAPT P10636 3/20 0.47
LMNA P02545 1/20 0.47
FAAH O00519 1/20 0.46
EPHX2 P34913 1/20 0.46
CHRNA7 P36544 1/20 0.44
RAB9A P51151 4/20 0.44
CCNA2 P20248 4/20 0.44
CDK2 P24941 4/20 0.44
ADORA3 P0DMS8 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
TUBB8B A6NNZ2 1/20 0.43
TUBB4A P04350 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20142465 0.90 CDK5 (0.52) NPC1MEN1KMT2ACDK5CDK5R1
SCHEMBL20141907 0.88 GSK3A (0.54) NPC1MEN1KMT2ACDK5CDK5R1
SCHEMBL20142502 0.88 MEN1 (0.64) NPC1MEN1KMT2ACDK5CDK5R1
SCHEMBL20142391 0.86 EPHX2 (0.48) NPC1MEN1KMT2ACDK5CDK5R1
SCHEMBL20142498 0.84 CCNA2 (0.52) NPC1MEN1KMT2ACDK5CDK5R1
SCHEMBL20142855 0.84 MEN1 (0.68) NPC1MEN1KMT2ACDK5CDK5R1
SCHEMBL20142189 0.84 CCNA2 (0.52) CDK5CDK5R1MAPTLMNACHRNA7
SCHEMBL20142496 0.81 MEN1 (0.66) NPC1MEN1KMT2ACDK5CDK5R1
SCHEMBL20142860 0.79 MEN1 (0.63) NPC1MEN1KMT2ACDK5CDK5R1
SCHEMBL20142426 0.79 MEN1 (0.63) NPC1MEN1KMT2ACDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089902-A1 DIAMINOTHIAZOLE COMPOUNDS, COMPOSITIONS AND METHODS OF USE APOGEE BIOTECHNOLOGY CORPORATION (US) 2018-05-17 WO claimed
WO-2018089902-A1 DIAMINOTHIAZOLE COMPOUNDS, COMPOSITIONS AND METHODS OF USE APOGEE BIOTECHNOLOGY CORPORATION (US) 2018-05-17 WO disclosed