SCHEMBL20142402

SCHEMBL20142402

CN(C)c1nc(Nc2ccc(F)cc2)sc1C(=O)c1ccc(Br)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.57
MEN1 O00255 4/20 0.57
KMT2A Q03164 4/20 0.57
RAB9A P51151 4/20 0.57
CCNA2 P20248 3/20 0.54
CDK2 P24941 3/20 0.54
CDK5 Q00535 7/20 0.53
CDK5R1 Q15078 7/20 0.53
MAPT P10636 6/20 0.46
LMNA P02545 3/20 0.46
TP53 P04637 2/20 0.46
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.46
DHODH Q02127 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
POLB P06746 1/20 0.44
GSK3A P49840 2/20 0.42
GSK3B P49841 2/20 0.42
MAPK14 Q16539 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20142409 0.90 GSK3A (0.53) NPC1MEN1KMT2ARAB9ACCNA2
SCHEMBL20142426 0.88 MEN1 (0.63) NPC1MEN1KMT2ARAB9ACCNA2
SCHEMBL20142192 0.82 CCNA2 (0.78) NPC1MEN1KMT2ARAB9ACCNA2
SCHEMBL20142179 0.78 GSK3A (0.53) NPC1MEN1KMT2ARAB9ACDK5
SCHEMBL20142391 0.78 EPHX2 (0.48) NPC1MEN1KMT2ARAB9ACCNA2
SCHEMBL20142841 0.78 MAPT (0.63) NPC1MEN1KMT2ARAB9ACCNA2
SCHEMBL20142502 0.77 MEN1 (0.64) NPC1MEN1KMT2ARAB9ACCNA2
SCHEMBL25609785 0.77 CDK5 (0.77) NPC1MEN1KMT2ARAB9ACCNA2
SCHEMBL20142267 0.77 GSK3A (0.51) NPC1MEN1KMT2ARAB9ACCNA2
SCHEMBL20142860 0.76 MEN1 (0.63) NPC1MEN1KMT2ACCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089902-A1 DIAMINOTHIAZOLE COMPOUNDS, COMPOSITIONS AND METHODS OF USE APOGEE BIOTECHNOLOGY CORPORATION (US) 2018-05-17 WO claimed
WO-2018089902-A1 DIAMINOTHIAZOLE COMPOUNDS, COMPOSITIONS AND METHODS OF USE APOGEE BIOTECHNOLOGY CORPORATION (US) 2018-05-17 WO disclosed