SCHEMBL20145157

SCHEMBL20145157

CN1CCC[C@@H](Nc2cnc(Cl)cn2)C1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KAT2B Q92831 12/20 0.52
BPTF Q12830 1/20 0.52
CCNK O75909 3/20 0.48
CDK12 Q9NYV4 3/20 0.48
IL1B P01584 5/20 0.46
NLRP3 Q96P20 1/20 0.46
CCNT1 O60563 1/20 0.42
CCNE1 P24864 1/20 0.42
CDK2 P24941 1/20 0.42
CDK9 P50750 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20145228 0.82 IL1B (0.54) KAT2BBPTFCCNKCDK12IL1B
SCHEMBL20145078 0.80 IL1B (0.46) KAT2BBPTFCCNKCDK12IL1B
SCHEMBL31333152 0.80 KAT2B (0.49) KAT2BBPTFCCNKCDK12IL1B
SCHEMBL20145184 0.78 IL1B (0.42) KAT2BBPTFIL1BNLRP3
SCHEMBL22654959 0.77 IL1B (0.61) KAT2BBPTFIL1BNLRP3
SCHEMBL22654958 0.77 IL1B (0.61) KAT2BBPTFIL1BNLRP3
SCHEMBL22655979 0.77 IL1B (0.61) KAT2BBPTFIL1BNLRP3
SCHEMBL23081193 0.76 BTK (0.46) KAT2BBPTFCCNKCDK12IL1B
SCHEMBL23081051 0.76 BTK (0.46) KAT2BBPTFCCNKCDK12IL1B
SCHEMBL22895690 0.75 CCNK (0.54) CCNKCDK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed