SCHEMBL20145078

SCHEMBL20145078

CN1CCCC(Nc2cnc(C(F)(F)F)cn2)C1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IL1B P01584 13/20 0.46
NLRP3 Q96P20 4/20 0.46
CCNK O75909 1/20 0.45
CDK12 Q9NYV4 1/20 0.45
KAT2B Q92831 6/20 0.43
BPTF Q12830 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20145184 0.90 IL1B (0.42) IL1BNLRP3KAT2BBPTF
SCHEMBL17031679 0.81 HCRTR1 (0.49) CCNKCDK12
SCHEMBL20144869 0.81 IL1B (0.55) IL1BNLRP3CCNKCDK12
SCHEMBL20145261 0.81 IL1B (0.55) IL1BNLRP3CCNKCDK12
SCHEMBL20145157 0.80 KAT2B (0.52) IL1BNLRP3CCNKCDK12KAT2B
SCHEMBL20145210 0.76 IL1B (0.49) IL1BNLRP3CCNKCDK12KAT2B
SCHEMBL20145228 0.73 IL1B (0.54) IL1BNLRP3CCNKCDK12KAT2B
SCHEMBL20145188 0.73 IL1B (0.43) IL1BNLRP3CCNKCDK12
SCHEMBL22877139 0.73 HCAR3 (0.45)
SCHEMBL23292323 0.72 CCNK (0.55) CCNKCDK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed