SCHEMBL20145188

SCHEMBL20145188

FC(F)(F)c1cnc(NC2CCCNC2)cn1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IL1B P01584 2/20 0.43
NLRP3 Q96P20 1/20 0.43
HCRTR1 O43613 2/20 0.43
IDH2 P48735 1/20 0.43
CCNK O75909 6/20 0.43
CDK12 Q9NYV4 6/20 0.43
CCNT1 O60563 5/20 0.43
CCNE1 P24864 5/20 0.43
CDK2 P24941 5/20 0.43
CDK9 P50750 5/20 0.43
CDK7 P50613 2/20 0.41
CCNH P51946 2/20 0.41
MNAT1 P51948 2/20 0.41
PIM1 P11309 1/20 0.41
IRAK4 Q9NWZ3 1/20 0.41
CHEK1 O14757 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22895360 0.92 PIK3CA (0.47) HCRTR1IDH2CCNKCDK12IRAK4
SCHEMBL17031679 0.84 HCRTR1 (0.49) HCRTR1CCNKCDK12
Trifluoroacetic Acid SCHEMBL28547919 0.83 HRH4 (0.54) HCRTR1CCNKCDK12IRAK4
Trifluoroacetic Acid SCHEMBL28547917 0.83 HRH4 (0.54) HCRTR1CCNKCDK12IRAK4
SCHEMBL20145185 0.80 IL1B (0.53) IL1BNLRP3HCRTR1IDH2CCNK
SCHEMBL22895689 0.78 IRAK4 (0.46) CCNKCDK12CCNT1CCNE1CDK2
Hydrochloric Acid SCHEMBL28546420 0.77 IRAK4 (0.45) CCNKCDK12CCNT1CCNE1CDK2
Hydrochloric Acid SCHEMBL28546424 0.77 IRAK4 (0.45) CCNKCDK12CCNT1CCNE1CDK2
SCHEMBL15440732 0.77 PRKCZ (0.51) CCNKCDK12CCNT1CCNE1CDK2
SCHEMBL25145695 0.75 HCRTR1 (0.40) HCRTR1IDH2CCNKCDK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed