SCHEMBL20145640

SCHEMBL20145640

Nc1ncc(-c2ccoc2)nc1-c1ccc(C(=O)NCc2ccccc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 17/20 0.68
ATR Q13535 2/20 0.50
HPGDS O60760 1/20 0.47
ROCK2 O75116 1/20 0.46
RPS6KA5 O75582 1/20 0.46
MAP4K4 O95819 1/20 0.46
PRKCG P05129 1/20 0.46
PRKACA P17612 1/20 0.46
RPS6KB1 P23443 1/20 0.46
AKT1 P31749 1/20 0.46
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
PRKX P51817 1/20 0.46
PRKCD Q05655 1/20 0.46
PRKG2 Q13237 1/20 0.46
ROCK1 Q13464 1/20 0.46
DYRK1A Q13627 1/20 0.46
PRKG1 Q13976 1/20 0.46
PKN2 Q16513 1/20 0.46
CDC42BPA Q5VT25 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16679751 0.81 MAPK1 (1.00) MAPK1
SCHEMBL16679747 0.81 MAPK1 (1.00) MAPK1
SCHEMBL20145591 0.81 MAPK1 (0.70) MAPK1HPGDSROCK2RPS6KA5MAP4K4
SCHEMBL20145662 0.80 MAPK1 (0.70) MAPK1
SCHEMBL16680183 0.76 MAPK1 (1.00) MAPK1HPGDSROCK2RPS6KA5MAP4K4
SCHEMBL3461899 0.75 ATR (0.68) MAPK1ATRHPGDS
SCHEMBL2934942 0.74 ALDH1A1 (0.53) MAPK1ATR
SCHEMBL1679733 0.73 LDHA (0.54) MAPK1ATRHPGDSROCK2MAP4K4
SCHEMBL3460691 0.72 LDHA (0.52) MAPK1ATRHPGDSMAP4K4PRKCG
SCHEMBL3459712 0.72 LDHA (0.63) ATRHPGDSMAP4K4PRKCGROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063143-B1 AMINOHETEROARYL BENZAMIDES AS KINASE INHIBITORS NOVARTIS AG (CH) 2018-05-16 EP disclosed