SCHEMBL20145923

SCHEMBL20145923

CC1=Nc2ccc(C)cc2CN1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
SMN1; SMN2 Q16637 4/20 0.36
GAA P10253 2/20 0.36
PARP10 Q53GL7 2/20 0.36
HTT P42858 2/20 0.36
PARP11 Q9NR21 1/20 0.36
HTR5A P47898 3/20 0.34
MAPT P10636 4/20 0.33
ALDH1A1 P00352 2/20 0.33
HSD17B10 Q99714 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
PARP1 P09874 1/20 0.33
HRH4 Q9H3N8 1/20 0.32
RAB9A P51151 5/20 0.32
FYN P06241 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
DYRK1B Q9Y463 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29419304 0.78
SCHEMBL1398128 0.76 NOS3 (0.39) PDE3BPDE3ASMN1; SMN2GAAHTR5A
SCHEMBL10354186 0.69 PDE3B (0.41) PDE3BPDE3ASMN1; SMN2GAAPARP10
SCHEMBL19142252 0.69 ADRA2A (0.36) PDE3BPDE3ASMN1; SMN2GAAPARP10
SCHEMBL13844803 0.69 PDE3B (0.41) PDE3BPDE3ATDP1
SCHEMBL19257866 0.69
SCHEMBL14294948 0.69 HTR5A (0.43) PDE3BPDE3AGAAPARP10PARP11
SCHEMBL2616770 0.68 PDE3B (0.41) PDE3BPDE3ASMN1; SMN2GAAPARP10
SCHEMBL2616781 0.65 PDE3B (0.39) PDE3BPDE3ASMN1; SMN2GAAPARP10
SCHEMBL30149404 0.65 PDE3B (0.39) PDE3BPDE3ASMN1; SMN2GAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3321261-A1 HEDGEHOG ANTAGONISTS HAVING ZINC BINDING MOIETIES Curis, Inc. (US) 2018-05-16 EP disclosed