SCHEMBL20145942

SCHEMBL20145942

CCCC(=O)c1cnc(=O)[nH]c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 1/20 0.42
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MMEL1 Q495T6 1/20 0.37
TLK2 Q86UE8 2/20 0.36
GABRA1 P14867 3/20 0.35
GABRG2 P18507 2/20 0.35
GABRB3 P28472 2/20 0.35
GABRA5 P31644 2/20 0.35
GABRA3 P34903 2/20 0.35
GABRA2 P47869 2/20 0.35
GABRB2 P47870 2/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRA4 P48169 1/20 0.35
GABRE P78334 1/20 0.35
GABRA6 Q16445 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9768122 0.76 MMEL1 (0.38) ALDH1A1MMEL1MME
SCHEMBL4649294 0.74 P4HA1 (0.43) ALDH1A1HPGDSMN1; SMN2MMEL1GABRA1
SCHEMBL20992124 0.73 HSD17B3 (0.46) HSD17B3ALDH1A1HPGDSMN1; SMN2L3MBTL1
SCHEMBL16891423 0.71 HSD17B3 (0.53) HSD17B3ALDH1A1HPGDSMN1; SMN2L3MBTL1
SCHEMBL27386679 0.68 HSD17B3 (0.53) HSD17B3HPGDSMN1; SMN2L3MBTL1STS
SCHEMBL9742618 0.68 MMEL1 (0.36) MMEL1MME
SCHEMBL11899972 0.67 NAPRT (0.56) HSD17B3ALDH1A1HPGDSMN1; SMN2L3MBTL1
SCHEMBL568662 0.67 HSD17B3 (0.52) HSD17B3HPGDSMN1; SMN2L3MBTL1STS
SCHEMBL29190968 0.67 TDP1 (0.63) HSD17B3ALDH1A1HPGDSMN1; SMN2L3MBTL1
SCHEMBL13838594 0.67 SMN1; SMN2 (0.56) HSD17B3HPGDSMN1; SMN2L3MBTL1GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3321261-B1 HEDGEHOG ANTAGONISTS HAVING ZINC BINDING MOIETIES CURIS INC (US) 2020-06-17 EP disclosed
EP-3321261-A1 HEDGEHOG ANTAGONISTS HAVING ZINC BINDING MOIETIES Curis, Inc. (US) 2018-05-16 EP disclosed