SCHEMBL4649294

SCHEMBL4649294

O=C(O)c1cnc(=O)[nH]c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P4HA1 P13674 2/20 0.43
P4HTM Q9NXG6 2/20 0.43
NOTUM Q6P988 1/20 0.43
MIF P14174 1/20 0.42
MMEL1 Q495T6 1/20 0.42
ALDH1A1 P00352 3/20 0.41
HSD17B10 Q99714 2/20 0.41
KDM4E B2RXH2 2/20 0.41
GABRP O00591 1/20 0.41
GABRD O14764 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRB1 P18505 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
GABRB2 P47870 1/20 0.41
GABRA4 P48169 1/20 0.41
GABRE P78334 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7232041 0.77 AXL (0.49) P4HA1P4HTMMMEL1ALDH1A1KDM4E
SCHEMBL9475882 0.77 P4HA1 (0.42) P4HA1P4HTMNOTUMMIFALDH1A1
SCHEMBL9742618 0.76 MMEL1 (0.36) MMEL1MME
SCHEMBL20145942 0.74 HSD17B3 (0.42) MMEL1ALDH1A1GABRPGABRDGABRA1
SCHEMBL5988807 0.69 GABRA1 (0.46) P4HTMMMEL1ALDH1A1HSD17B10KDM4E
SCHEMBL4886683 0.68 ALDH1A1 (0.58) P4HA1P4HTMMIFALDH1A1HSD17B10
SCHEMBL4600260 0.67 ALDH1A1 (0.52) P4HA1P4HTMMIFALDH1A1HSD17B10
Benzamide SCHEMBL23248639 0.65 PARP1 (0.48) MMEL1ALDH1A1HSD17B10KDM4ECYP1A2
SCHEMBL29864 0.65
SCHEMBL4422067 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1675834-A4 COMPOUNDS, COMPOSITIONS, AND METHODS CYTOKINETICS INC (US) 2008-08-27 EP claimed
EP-1675834-A1 COMPOUNDS, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2006-07-05 EP claimed
WO-2005037799-A1 COMPOUNDS, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2005-04-28 WO claimed
CN-107250110-A The noval chemical compound of (RET) inhibitor is reset as transfection 葛兰素史克知识产权发展有限公司 2017-10-13 CN disclosed
WO-2009114470-A2 TETRAHYDROINDOLE AND TETRAHDYROINDAZOLE AS HSP90 INHIBITORS CONTAINING A ZINC BINDING MOIETY CURIS, INC. (US) 2009-09-17 WO disclosed