SCHEMBL2014620

SCHEMBL2014620

COC(=O)c1ccc([N+](=O)[O-])c(OCC(=O)c2ccccc2)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.66
MEN1 O00255 2/20 0.66
KMT2A Q03164 2/20 0.66
MAPT P10636 3/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
AR P10275 1/20 0.54
PELP1 Q8IZL8 1/20 0.54
KDM4E B2RXH2 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
HPGD P15428 1/20 0.48
CYP2C19 P33261 1/20 0.48
AKR1C3 P42330 2/20 0.48
AKR1C2 P52895 2/20 0.48
AKR1C1 Q04828 2/20 0.48
AKR1C4 P17516 1/20 0.48
VCAM1 P19320 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2011302 0.89 AR (0.53) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL2978081 0.85 AR (0.58) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL29979942 0.85 AR (0.58) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL527105 0.84 MYC (0.59) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL30082879 0.84 MYC (0.59) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL30669432 0.84 AR (0.57) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL8570002 0.84 AR (0.57) ALDH1A1KMT2AMAPTARPELP1
SCHEMBL10318922 0.84 AR (0.57) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL221362 0.82 AR (0.61) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL2013298 0.81 ALDH1A1 (0.71) ALDH1A1MEN1KMT2AMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073273-A1 BENZOXAZINE ARYL SULFONAMIDE DERIVATIVES AS KV1.3 MODULATORS EVOTEC AG (DE) 2011-06-23 WO disclosed
WO-2011073276-A1 BENZOXAZINE ARYL SULFONAMIDE DERIVATIVES AS KV1.3 MODULATORS EVOTEC AG (DE) 2011-06-23 WO disclosed