SCHEMBL2014762

SCHEMBL2014762

O=C(NCc1cccc(C(F)(F)F)c1)C1CCC(c2ccccc2)N(S(=O)(=O)c2ccccc2)C1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.56
KDM4E B2RXH2 1/20 0.53
RAB9A P51151 2/20 0.51
NPC1 O15118 1/20 0.51
CCR2 P41597 2/20 0.49
TSHR P16473 1/20 0.49
PKM P14618 2/20 0.48
LMNA P02545 1/20 0.48
P2RX7 Q99572 1/20 0.47
MMP1 P03956 1/20 0.46
ADAM17 P78536 1/20 0.46
PLA2G1B P04054 1/20 0.45
ATG4B Q9Y4P1 1/20 0.45
NR1H2 P55055 1/20 0.45
NR1H3 Q13133 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12628160 1.00 KMT2A (0.56) KMT2AKDM4ERAB9ANPC1CCR2
SCHEMBL2017811 0.89 ALDH1A1 (0.50) KMT2ARAB9ACCR2PKMP2RX7
SCHEMBL12628167 0.89 ALDH1A1 (0.50) KMT2ARAB9ACCR2PKMP2RX7
SCHEMBL2013288 0.89 PKM (0.49) KMT2ARAB9ATSHRPKMLMNA
SCHEMBL12628169 0.89 PKM (0.49) KMT2ARAB9ATSHRPKMLMNA
SCHEMBL2011504 0.88 ALDH1A1 (0.54) KMT2ARAB9APKM
SCHEMBL12628159 0.88 ALDH1A1 (0.54) KMT2ARAB9APKM
SCHEMBL12629088 0.87 KMT2A (0.56) KMT2ARAB9APKM
SCHEMBL2011797 0.87 KMT2A (0.56) KMT2ARAB9APKM
SCHEMBL2015115 0.85 ALDH1A1 (0.51) KMT2ATSHRPKMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073269-A1 PIPERIDINE ARYL SULFONAMIDE DERIVATIVES AS KV1.3 MODULATORS EVOTEC AG (DE) 2011-06-23 WO claimed