SCHEMBL20149928

SCHEMBL20149928

CNC1CCN(c2ccccc2C#N)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 2/20 0.44
DRD4 P21917 5/20 0.43
DRD2 P14416 4/20 0.43
GRM5 P41594 1/20 0.43
MTOR P42345 4/20 0.42
RPTOR Q8N122 4/20 0.42
MLST8 Q9BVC4 4/20 0.42
DRD3 P35462 3/20 0.42
CHRM4 P08173 1/20 0.41
KDM1A O60341 1/20 0.41
CYP3A4 P08684 2/20 0.41
AR P10275 1/20 0.41
HTR7 P34969 1/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
CDC42BPB Q9Y5S2 1/20 0.40
PHGDH O43175 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20149778 0.83 DRD4 (0.43) KDM4EALDH1A1DRD4DRD2GRM5
SCHEMBL13176022 0.81 MEN1 (0.59) KDM4EALDH1A1DRD4DRD2GRM5
SCHEMBL31042527 0.79 DRD4 (0.51) KDM4EALDH1A1DRD4DRD2GRM5
SCHEMBL18840246 0.79 ROCK2 (0.45) KDM4EALDH1A1MTORRPTORMLST8
SCHEMBL3088832 0.78 DRD4 (0.54) KDM4EALDH1A1DRD4DRD2GRM5
SCHEMBL2261269 0.78 KDM4E (0.47) KDM4EALDH1A1DRD4DRD2GRM5
SCHEMBL8693892 0.78 ADRB1 (0.50) KDM4EALDH1A1DRD2DRD3CYP2D6
SCHEMBL20140119 0.78 GRM5 (0.49) KDM4EALDH1A1DRD4DRD2GRM5
SCHEMBL7714987 0.78 KDM4E (0.44) KDM4EALDH1A1DRD4DRD2GRM5
SCHEMBL20756875 0.77 KDM4E (0.44) KDM4EALDH1A1DRD4DRD2GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089499-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed