SCHEMBL2015023

SCHEMBL2015023

O=C(Nc1ccccc1)C1CCC(c2ccc(F)cc2)N(S(=O)(=O)c2ccccc2)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.48
TRPA1 O75762 1/20 0.48
ALDH1A1 P00352 4/20 0.48
KMT2A Q03164 3/20 0.48
RAB9A P51151 1/20 0.48
MEN1 O00255 1/20 0.47
FAAH O00519 1/20 0.47
GAA P10253 2/20 0.47
MAPT P10636 2/20 0.47
LMNA P02545 1/20 0.47
HTT P42858 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
CHRNB2 P17787 1/20 0.46
CHRNB4 P30926 1/20 0.46
CHRNA3 P32297 1/20 0.46
CHRNA4 P43681 1/20 0.46
BRD4 O60885 1/20 0.45
TP53 P04637 1/20 0.45
TSHR P16473 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12628296 1.00 DPP4 (0.48) DPP4TRPA1ALDH1A1KMT2ARAB9A
SCHEMBL12628166 0.96 ALDH1A1 (0.51) DPP4ALDH1A1KMT2ARAB9AMEN1
SCHEMBL2012495 0.96 ALDH1A1 (0.51) DPP4ALDH1A1KMT2ARAB9AMEN1
SCHEMBL12629075 0.92 ALDH1A1 (0.57) ALDH1A1KMT2ARAB9AMEN1FAAH
SCHEMBL2013828 0.92 ALDH1A1 (0.57) ALDH1A1KMT2ARAB9AMEN1FAAH
SCHEMBL2010268 0.88 TSHR (0.48) ALDH1A1KMT2ARAB9AMEN1GAA
SCHEMBL12628945 0.88 TSHR (0.48) ALDH1A1KMT2ARAB9AMEN1GAA
SCHEMBL12628292 0.84 KMT2A (0.55) ALDH1A1KMT2AMEN1TP53TSHR
SCHEMBL2015653 0.84 KMT2A (0.55) ALDH1A1KMT2AMEN1TP53TSHR
SCHEMBL12628165 0.83 SMN1; SMN2 (0.53) ALDH1A1KMT2ARAB9AMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073269-A1 PIPERIDINE ARYL SULFONAMIDE DERIVATIVES AS KV1.3 MODULATORS EVOTEC AG (DE) 2011-06-23 WO claimed