SCHEMBL2054419

SCHEMBL2054419

COc1cc(C(=O)N(C)[C@H](CCNC(=O)c2cccn2C)Cc2ccccc2)c2nc(C)ccc2c1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.58
HCRTR2 O43614 2/20 0.58
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
ALDH1A1 P00352 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRK1 P41145 1/20 0.35
HRH3 Q9Y5N1 3/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PADI4 Q9UM07 2/20 0.33
PYGL P06737 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2013457 1.00 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9AALDH1A1
SCHEMBL2015171 0.89 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9AALDH1A1
SCHEMBL2017008 0.89 HCRTR1 (0.56) HCRTR1HCRTR2NPC1RAB9AALDH1A1
SCHEMBL2012853 0.87 HCRTR1 (0.59) HCRTR1HCRTR2NPC1RAB9AALDH1A1
SCHEMBL13139077 0.83 HCRTR1 (0.75) HCRTR1HCRTR2NPC1RAB9AALDH1A1
SCHEMBL2016967 0.83 HCRTR1 (0.55) HCRTR1HCRTR2NPC1RAB9AALDH1A1
SCHEMBL2053397 0.83 HCRTR1 (0.55) HCRTR1HCRTR2NPC1RAB9AALDH1A1
SCHEMBL2015020 0.82 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2010990 0.82 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2011939 0.82 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed