SCHEMBL20153326

SCHEMBL20153326

CCOC(=O)CC(c1ccc(OC)nc1)n1ccc(Br)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.40
ALDH1A1 P00352 5/20 0.40
HTT P42858 1/20 0.40
OXTR P30559 1/20 0.39
MAPT P10636 4/20 0.37
LMNA P02545 1/20 0.37
JMJD6 Q6NYC1 1/20 0.35
FFAR1 O14842 1/20 0.34
RAB9A P51151 2/20 0.33
NNMT P40261 1/20 0.33
FGFR2 P21802 1/20 0.33
FGFR3 P22607 1/20 0.33
KMT2A Q03164 5/20 0.33
MEN1 O00255 4/20 0.33
POLB P06746 3/20 0.33
GAA P10253 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KCNK3 O14649 1/20 0.32
NPC1 O15118 1/20 0.32
PABPC1 P11940 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20153360 0.86 OXTR (0.34) KDM4EALDH1A1OXTRMAPTRAB9A
SCHEMBL20153309 0.83 KDM4E (0.35) KDM4EALDH1A1HTTOXTRMAPT
SCHEMBL21311520 0.83 ITGB3 (0.37) KDM4EALDH1A1HTTOXTRMAPT
SCHEMBL21311585 0.82 OXTR (0.36) KDM4EALDH1A1HTTOXTRMAPT
SCHEMBL20153308 0.82 KDM4E (0.35) KDM4EALDH1A1HTTOXTRMAPT
SCHEMBL20153325 0.81 FYN (0.41) OXTRJMJD6KMT2AMEN1
SCHEMBL20153458 0.81 OXTR (0.35) KDM4EALDH1A1HTTOXTRMAPT
SCHEMBL23677937 0.80 JMJD6 (0.36) KDM4EALDH1A1HTTOXTRMAPT
SCHEMBL21311521 0.77 ITGB3 (0.38) ITGB3ITGAV
SCHEMBL20153330 0.76 OXTR (0.35) KDM4EALDH1A1HTTOXTRJMJD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538525-B1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2022-06-22 EP disclosed
WO-2018089353-A1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed