SCHEMBL20153412

SCHEMBL20153412

Cc1ncc(C(CC(=O)OC(C)(C)C)N/C=C\C(=N)CCCc2ccc3c(n2)NCCCC3)cn1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.49
ITGB3 P05106 17/20 0.49
ITGB6 P18564 9/20 0.45
ITGB5 P18084 7/20 0.43
ITGB8 P26012 7/20 0.43
ITGA2B P08514 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20153505 0.90 ITGB3 (0.53) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL20153504 0.88 ITGB3 (0.62) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL24521878 0.88 ITGAV (0.57) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL24521828 0.86 ITGAV (0.60) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL24521933 0.85 ITGAV (0.50) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL24521991 0.84 ITGB3 (0.60) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL24521913 0.82 ITGB3 (0.63) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL24521903 0.81 ITGAV (0.61) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL20153461 0.81 ITGAV (0.59) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL20153385 0.79 ITGAV (0.64) ITGAVITGB3ITGB6ITGB5ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089353-A1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed