SCHEMBL20153435

SCHEMBL20153435

CC(NS(=O)(=O)c1cnc(N2CCN3C[C@H](O)C[C@H]3C2)s1)c1ccccc1-c1cncn1CCc1ccc(F)cc1

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16719037 1.00 HSP90AA1 (0.32) HSP90AA1HSP90AB1
SCHEMBL16719040 1.00 HSP90AA1 (0.32) HSP90AA1HSP90AB1
SCHEMBL20170514 0.90 KCNH2 (0.32) HSP90AA1HSP90AB1
SCHEMBL16719021 0.87
SCHEMBL16730819 0.86 SLC1A2 (0.35) HSP90AA1HSP90AB1
SCHEMBL20169617 0.81 ADRA2C (0.30)
SCHEMBL16718973 0.81 ADRA2C (0.30)
SCHEMBL16720946 0.81 CYP11B2 (0.32)
SCHEMBL16719019 0.80 SCN9A (0.31)
SCHEMBL16719058 0.78 SLC1A2 (0.34) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068391-B1 ARYL LINKED IMIDAZOLE AND TRIAZOLE DERIVATIVES AND METHODS OF USE THEREOF FOR IMPROVING THE PHARMACOKINETICS OF A DRUG MERCK SHARP & DOHME (US) 2018-05-23 EP claimed
US-9975888-B2 Aryl linked imidazole and triazole derivatives and methods of use thereof for improving the pharmacokinetics of a drug MERCK SHARP & DOHME CORP. (US) 2018-05-22 US claimed
EP-3068391-B1 ARYL LINKED IMIDAZOLE AND TRIAZOLE DERIVATIVES AND METHODS OF USE THEREOF FOR IMPROVING THE PHARMACOKINETICS OF A DRUG MERCK SHARP & DOHME (US) 2018-05-23 EP disclosed