SCHEMBL20153524

SCHEMBL20153524

CCOC(=O)[C@@H]1CCC2c3ccc(C)cc3N(C(=O)OC(C)C)CC21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.35
ALOX12 P18054 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 4/20 0.34
HPGD P15428 1/20 0.34
CHRNA1 P02708 1/20 0.34
CHRNG P07510 1/20 0.34
ITGA5 P08648 1/20 0.34
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
SLC6A2 P23975 1/20 0.34
CHRNB4 P30926 1/20 0.34
SLC6A4 P31645 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
SLC6A3 Q01959 1/20 0.34
CHRND Q07001 1/20 0.34
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20153621 0.90 MEN1 (0.36) GAAALDH1A1CA12CA1CA2
SCHEMBL20131503 0.77 CA12 (0.32) ALDH1A1CA12CA1CA2CA9
SCHEMBL20131490 0.77 MEN1 (0.35) GAAALDH1A1CA12CA1CA2
SCHEMBL20131461 0.74 RORC (0.39) SMN1; SMN2ALDH1A1
SCHEMBL22297669 0.72 HSD17B1 (0.45) CA12CA1CA2CA9KMT2A
SCHEMBL22297671 0.72 HSD17B1 (0.45) CA12CA1CA2CA9KMT2A
SCHEMBL22297656 0.72 HSD17B1 (0.45) CA12CA1CA2CA9KMT2A
SCHEMBL30636993 0.64 HTR2A (0.49) HPGDCA12CA1CA2CA9
SCHEMBL6081536 0.61 MAPT (0.47) GAAALDH1A1HPGDSLC6A4SLC6A3
SCHEMBL16306571 0.59 PPM1B (0.40) ALDH1A1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089402-A1 TRICYCLIC SULFONES AS ROR GAMMA MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed