SCHEMBL20153719

SCHEMBL20153719

C=Cc1cccnc1N(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.37
ALDH1A1 P00352 2/20 0.37
POLB P06746 2/20 0.37
TRIM24 O15164 1/20 0.34
TRIM33 Q9UPN9 1/20 0.34
SYK P43405 1/20 0.33
LMNA P02545 3/20 0.33
HIF1A Q16665 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C9 P11712 2/20 0.33
MAPK1 P28482 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
MAPT P10636 3/20 0.32
HTT P42858 2/20 0.32
APP P05067 1/20 0.31
SNCA P37840 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
MITF O75030 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18726709 0.80 KDM4E (0.37) KDM4EALDH1A1POLBTRIM24TRIM33
SCHEMBL29954331 0.80 TRIM24 (0.52) KDM4EALDH1A1POLBTRIM24TRIM33
SCHEMBL12253115 0.80 TRIM24 (0.52) KDM4EALDH1A1POLBTRIM24TRIM33
SCHEMBL9000291 0.76 KDM4E (0.38) KDM4EALDH1A1POLBTRIM24TRIM33
SCHEMBL6493230 0.74 GRM5 (0.50) KDM4EALDH1A1APPSNCA
SCHEMBL14918245 0.74 KDM4E (0.41) KDM4EALDH1A1POLBSYKLMNA
SCHEMBL16343065 0.72
SCHEMBL935465 0.72
SCHEMBL761273 0.72 ALDH1A1 (0.41) KDM4EALDH1A1POLBSYKLMNA
SCHEMBL20586643 0.72 CXCR4 (0.40) ALDH1A1POLBTRIM24TRIM33CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538525-B1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2022-06-22 EP disclosed
EP-3538519-B1 INDAZOLE DERIVATIVES AS ALPHA V INTEGRIN ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2021-07-28 EP disclosed
WO-2018089357-A1 INDAZOLE DERIVATIVES AS αV INTEGRIN ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed
CN-106215894-A A kind of preparation method of lysine purification adsorbent 王琪宇 2016-12-14 CN disclosed