SCHEMBL2015482

SCHEMBL2015482

CC1(C)CC(C)(C)c2cc(-c3cccc(N4CCN(C(=O)O)CC4)n3)ccc21

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RARA P10276 2/20 0.50
RARB P10826 2/20 0.50
CNR1 P21554 15/20 0.44
PIM1 P11309 1/20 0.44
PIM2 Q9P1W9 1/20 0.44
RARG P13631 2/20 0.39
FAAH O00519 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12959456 0.93 RARB (0.59) RARARARBCNR1PIM1PIM2
SCHEMBL2016042 0.85 CKS1B (0.48) RARARARBCNR1
SCHEMBL27973420 0.85 RARA (0.47) RARARARBCNR1PIM1PIM2
SCHEMBL27872046 0.84 RARA (0.46) RARARARBCNR1PIM1PIM2
SCHEMBL2039478 0.81 HTR3E (0.46) RARARARBPIM1PIM2
SCHEMBL2018037 0.79 RARB (0.56) RARARARBCNR1PIM1PIM2
SCHEMBL2015994 0.79 RARA (0.50) RARARARBCNR1RARG
SCHEMBL12959457 0.79 RARB (0.54) RARARARBCNR1PIM1PIM2
SCHEMBL8514041 0.79 RARB (0.46) RARARARBPIM1PIM2RARG
SCHEMBL2015316 0.78 HTR1A (0.45) RARARARBCNR1PIM1PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102666489-B Sphingosine kinase inhibitors MERCK PATENT GMBH 2014-07-23 CN disclosed
EP-2513057-A1 SPHINGOSINE KINASE INHIBITORS Merck Patent GmbH (DE) 2012-10-24 EP disclosed
CN-102666489-A Sphingosine kinase inhibitors MERCK PATENT GMBH 2012-09-12 CN disclosed
WO-2011072791-A1 SPHINGOSINE KINASE INHIBITORS MERCK PATENT GMBH (DE) 2011-06-23 WO disclosed