SCHEMBL20154910

SCHEMBL20154910

Cc1cc(Nc2ncc(Br)c(NC3CCN(C(=O)OC(C)(C)C)CC3)n2)no1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 5/20 0.48
AXL P30530 1/20 0.46
MERTK Q12866 1/20 0.46
SYK P43405 3/20 0.43
GPR119 Q8TDV5 2/20 0.43
AURKA O14965 1/20 0.43
AURKB Q96GD4 1/20 0.43
NSD2 O96028 1/20 0.42
KDM1A O60341 1/20 0.42
EHMT2 Q96KQ7 1/20 0.42
RCOR1 Q9UKL0 1/20 0.42
CCNK O75909 1/20 0.42
CCNA2 P20248 1/20 0.42
CDK2 P24941 1/20 0.42
CCND3 P30281 1/20 0.42
CDK9 P50750 1/20 0.42
CDK6 Q00534 1/20 0.42
DNMT3A Q9Y6K1 1/20 0.42
ALDH1A1 P00352 1/20 0.41
ALK Q9UM73 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20154980 0.85 IGF1R (0.57) IGF1RSYKGPR119AURKAAURKB
SCHEMBL20154906 0.78 ALDH1A1 (0.51) GPR119NSD2KDM1AEHMT2RCOR1
SCHEMBL20154982 0.78 ALDH1A1 (0.49) GPR119NSD2KDM1AEHMT2RCOR1
SCHEMBL4071068 0.78 SYK (0.51) IGF1RSYKAURKAAURKBCCNK
SCHEMBL20154930 0.78 IGF1R (0.51) IGF1RSYKGPR119AURKAAURKB
SCHEMBL6832459 0.76 SYK (0.57) IGF1RSYKGPR119AURKAAURKB
SCHEMBL21299894 0.75 SYK (0.42) IGF1RMERTKSYKGPR119AURKA
SCHEMBL11346537 0.75 IGF1R (0.71) IGF1R
SCHEMBL4067722 0.74 SYK (0.58) IGF1RMERTKSYKGPR119AURKA
SCHEMBL11932348 0.73 IGF1R (0.54) IGF1RSYKGPR119DNMT3AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3530656-B1 2-SUBSTITUTED AROMATIC RING-PYRIMIDINE DERIVATIVE, AND PREPARATION AND APPLICATION THEREOF UNIV ZHEJIANG (CN) 2022-01-05 EP disclosed
WO-2018086547-A1 2-SUBSTITUTED AROMATIC RING-PYRIMIDINE DERIVATIVE, AND PREPARATION AND APPLICATION THEREOF 浙江大学 2018-05-17 WO disclosed