SCHEMBL20154945

SCHEMBL20154945

CCNS(=O)(=O)c1ccc(Oc2ccc(F)cc2F)c(Br)c1

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 6/20 0.62
ALDH1A1 P00352 2/20 0.53
KMT2A Q03164 1/20 0.47
PKM P14618 1/20 0.45
MEP1B Q16820 1/20 0.44
SLC22A12 Q96S37 1/20 0.43
GLA P06280 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
BRD4 O60885 1/20 0.41
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16650857 0.84 EPAS1 (0.67) EPAS1BRD4PTGS1PTGS2
SCHEMBL20155313 0.83 MEP1B (0.43) EPAS1ALDH1A1MEP1BSLC22A12BRD4
SCHEMBL16651328 0.81 EPAS1 (0.71) EPAS1BRD4PTGS1PTGS2
SCHEMBL30306252 0.81 EPAS1 (0.71) EPAS1BRD4PTGS1PTGS2
SCHEMBL16650802 0.80 EPAS1 (0.72) EPAS1BRD4PTGS1PTGS2
SCHEMBL15067831 0.78 EPAS1 (0.66) EPAS1BRD4PTGS1PTGS2
SCHEMBL3006563 0.78 ALDH1A1 (0.63) ALDH1A1KMT2AMEP1BSMN1; SMN2
SCHEMBL20155326 0.78 ALDH1A1 (0.59) ALDH1A1KMT2APKMSMN1; SMN2
SCHEMBL16555815 0.76 EPAS1 (1.00) EPAS1
SCHEMBL16333294 0.76 BRD4 (0.57) EPAS1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed