SCHEMBL20155313

SCHEMBL20155313

CCNS(=O)(=O)c1ccc(Oc2ccc(F)cc2F)c(B(O)O)c1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MEP1B Q16820 1/20 0.43
ALDH1A1 P00352 2/20 0.42
EPAS1 Q99814 1/20 0.42
SLC22A12 Q96S37 1/20 0.41
TSHR P16473 1/20 0.40
BRD4 O60885 5/20 0.40
IDH2 P48735 1/20 0.39
PTGER3 P43115 1/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
PNMT P11086 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20154945 0.83 EPAS1 (0.62) MEP1BALDH1A1EPAS1SLC22A12BRD4
SCHEMBL16651491 0.77 BRD4 (0.55) BRD4
SCHEMBL3203639 0.74 MEP1B (0.46) MEP1BALDH1A1
SCHEMBL20155378 0.73 TRPA1 (0.35) BRD4
SCHEMBL16195782 0.72 ALDH1A1 (0.54) ALDH1A1TSHRPNMT
SCHEMBL29956502 0.72 ALDH1A1 (0.54) ALDH1A1TSHRPNMT
SCHEMBL28505143 0.72 ENPP2 (0.48) ALDH1A1
SCHEMBL13595012 0.70 GBA1 (0.56) ALDH1A1BRD4
SCHEMBL6290082 0.69 ALDH1A1 (0.68) MEP1BALDH1A1TSHR
SCHEMBL15068027 0.69 SCN8A (0.46) EPAS1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed