SCHEMBL20154979

SCHEMBL20154979

CC(C)(C)OC(=O)N1CCC(CNc2nc(N)ncc2Br)CC1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCDIN3D Q7Z5W3 1/20 0.53
SYK P43405 1/20 0.50
GPR119 Q8TDV5 6/20 0.48
KDM4E B2RXH2 2/20 0.47
PKM P14618 1/20 0.47
IDO1 P14902 2/20 0.47
TDO2 P48775 1/20 0.47
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43
CDK5 Q00535 1/20 0.43
CDK5R1 Q15078 1/20 0.43
PRMT5 O14744 1/20 0.42
FAAH O00519 1/20 0.42
MAPT P10636 1/20 0.41
FPR3 P25089 1/20 0.41
FPR2 P25090 1/20 0.41
TRPV1 Q8NER1 1/20 0.40
TGFBR1 P36897 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17764590 0.88 BCDIN3D (0.51) BCDIN3DSYKGPR119KDM4EPKM
SCHEMBL20154982 0.84 ALDH1A1 (0.49) GPR119CCNA2CDK2MAPT
SCHEMBL20155228 0.84 KDM4E (0.53) BCDIN3DSYKGPR119KDM4EPKM
SCHEMBL20155296 0.82 IRAK1 (0.60) BCDIN3DSYKGPR119
SCHEMBL2460443 0.82 IDO1 (0.54) BCDIN3DSYKGPR119KDM4EPKM
SCHEMBL2460448 0.82 IDO1 (0.54) BCDIN3DSYKGPR119KDM4EPKM
SCHEMBL2463486 0.82 IDO1 (0.54) BCDIN3DSYKGPR119KDM4EPKM
SCHEMBL620235 0.82 IDO1 (0.53) BCDIN3DSYKGPR119KDM4EPKM
SCHEMBL3779057 0.80 KDM4E (0.53) BCDIN3DSYKGPR119KDM4EPKM
SCHEMBL20155297 0.80 SYK (0.49) BCDIN3DSYKGPR119KDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3530656-B1 2-SUBSTITUTED AROMATIC RING-PYRIMIDINE DERIVATIVE, AND PREPARATION AND APPLICATION THEREOF UNIV ZHEJIANG (CN) 2022-01-05 EP disclosed
WO-2018086547-A1 2-SUBSTITUTED AROMATIC RING-PYRIMIDINE DERIVATIVE, AND PREPARATION AND APPLICATION THEREOF 浙江大学 2018-05-17 WO disclosed