SCHEMBL20155048

SCHEMBL20155048

CC1(C)OB(c2cc(N)c(C(N)=O)cc2Oc2ccc(F)cc2F)OC1(C)C

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.42
HSPB1 P04792 2/20 0.36
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
CARM1 Q86X55 1/20 0.34
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
SCN4A P35499 1/20 0.33
MAPT P10636 1/20 0.33
KEAP1 Q14145 1/20 0.33
SCN8A Q9UQD0 1/20 0.32
SCN10A Q9Y5Y9 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155120 0.85 ALDH1A1 (0.40) BRD4HSPB1ALDH1A1PTGS2
SCHEMBL15069672 0.79 HSPB1 (0.39) BRD4HSPB1ALDH1A1PTGS2
SCHEMBL29533045 0.79 HSPB1 (0.39) BRD4HSPB1ALDH1A1PTGS2
SCHEMBL22858968 0.77 HSPB1 (0.39) BRD4HSPB1ALDH1A1GAAMAPT
SCHEMBL20154948 0.75 EPAS1 (0.46) BRD4HSPB1LMNAHTTALDH1A1
SCHEMBL21191032 0.75 BRD4 (0.45) BRD4ALDH1A1GAAL3MBTL1MAPT
SCHEMBL31073743 0.75 HSPB1 (0.38) BRD4HSPB1CARM1PTGS2
SCHEMBL20155663 0.75 HSPB1 (0.36) HSPB1ALDH1A1PTGS2
SCHEMBL15069481 0.73 BRD4 (0.48) BRD4HSPB1PTGS2
SCHEMBL21904915 0.73 HSPB1 (0.39) BRD4HSPB1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed