SCHEMBL20155072

SCHEMBL20155072

CC1(C)OB(c2cc(N)ccc2Oc2ccccc2F)OC1(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
HSPB1 P04792 1/20 0.39
CARM1 Q86X55 3/20 0.36
PRMT6 Q96LA8 3/20 0.36
LPL P06858 2/20 0.34
LIPG Q9Y5X9 2/20 0.34
EGFR P00533 1/20 0.34
RHEB Q15382 1/20 0.33
JAK2 O60674 1/20 0.32
BTK Q06187 1/20 0.32
PIK3CG P48736 1/20 0.32
ROCK1 Q13464 1/20 0.32
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 1/20 0.31
ESR1 P03372 1/20 0.31
HTR1A P08908 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A3 Q01959 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29533045 0.90 HSPB1 (0.39) HSPB1LPLLIPGEGFRALDH1A1
SCHEMBL15069672 0.90 HSPB1 (0.39) HSPB1LPLLIPGEGFRALDH1A1
SCHEMBL21904778 0.87 JAK2 (0.34) LPLLIPGEGFRJAK2BTK
SCHEMBL20155409 0.85 SLC6A2 (0.39) EGFRALDH1A1SLC6A2SLC6A3
SCHEMBL30748970 0.84 LPL (0.40) MEN1KMT2AHSPB1CARM1PRMT6
SCHEMBL20160238 0.83 SLC6A4 (0.38) LPLLIPGEGFRBTKPIK3CG
SCHEMBL21904898 0.83 LPL (0.41) MEN1KMT2AHSPB1CARM1PRMT6
SCHEMBL15328685 0.82 BRD4 (0.40) MEN1KMT2ALPLLIPGMAPT
SCHEMBL20155416 0.82 SLC6A2 (0.40) LPLLIPGEGFRMAPTALDH1A1
SCHEMBL20155469 0.79 KDM4E (0.42) LPLLIPGALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed