SCHEMBL20155409

SCHEMBL20155409

CC1(C)OB(c2cc(N)ccc2Oc2ccc(Cl)cc2F)OC1(C)C

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
KCNH2 Q12809 1/20 0.39
SLC6A3 Q01959 1/20 0.39
EGFR P00533 3/20 0.39
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
LIPE Q05469 1/20 0.32
PTGS2 P35354 4/20 0.32
PTGS1 P23219 1/20 0.32
SCN9A Q15858 1/20 0.31
PPARG P37231 2/20 0.31
PPARA Q07869 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15069672 0.87 HSPB1 (0.39) EGFRALDH1A1PTGS2
SCHEMBL29533045 0.87 HSPB1 (0.39) EGFRALDH1A1PTGS2
SCHEMBL20155072 0.85 MEN1 (0.40) SLC6A2SLC6A3EGFRALDH1A1
SCHEMBL20155354 0.83 MAPT (0.44) SLC6A4KCNH2EGFRALDH1A1HPGD
SCHEMBL20155416 0.82 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3EGFRALDH1A1
SCHEMBL20155393 0.82 KDM4E (0.42) EGFRALDH1A1HPGDSCN9A
SCHEMBL21904908 0.81 HTR2A (0.41) SLC6A4KCNH2EGFRALDH1A1POLB
SCHEMBL21904778 0.80 JAK2 (0.34) SLC6A2EGFRPOLB
SCHEMBL20160238 0.79 SLC6A4 (0.38) SLC6A2SLC6A4SLC6A3EGFRPTGS2
SCHEMBL21904898 0.78 LPL (0.41) SLC6A4KCNH2EGFRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed
US-9249355-B2 Liquid-crystal displays having homeotropic alignment MERCK PATENT GMBH (DE) 2016-02-02 US disclosed