SCHEMBL20155112

SCHEMBL20155112

O=c1[nH]ccc2nn(Cc3ccccc3)cc12

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.52
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
MAPT P10636 1/20 0.41
KDM4C Q9H3R0 2/20 0.40
MPO P05164 1/20 0.40
PRKACA P17612 1/20 0.40
PRKACG P22612 1/20 0.40
PRKACB P22694 1/20 0.40
HTR2C P28335 1/20 0.40
P2RX7 Q99572 1/20 0.39
PLK1 P53350 1/20 0.39
CCNK O75909 1/20 0.39
CDK12 Q9NYV4 1/20 0.39
PARP1 P09874 2/20 0.38
KMT2A Q03164 1/20 0.38
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
MGLL Q99685 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22206944 0.82 CCNK (0.45) ADORA3MAPTCCNKCDK12KMT2A
SCHEMBL20155602 0.76 IP6K1 (0.40) ADORA3MAPTKDM4CP2RX7PARP1
SCHEMBL7479263 0.75 MAPT (0.52) ADORA3ADORA2AADORA1MAPTPARP1
SCHEMBL20155109 0.74 ADORA3 (0.56) ADORA3ADORA2AADORA1MAPTHTR2C
SCHEMBL20155563 0.72 CNR2 (0.42) MPO
SCHEMBL11155364 0.72 MPO (0.46) ADORA3ADORA2AADORA1MAPTMPO
SCHEMBL4792680 0.72 MPO (0.46) ADORA3ADORA2AADORA1MPOHTR2C
SCHEMBL1169684 0.72 MPO (0.46) ADORA3ADORA2AADORA1MPOHTR2C
SCHEMBL4791000 0.71 ADORA3 (0.45) ADORA3ADORA2AADORA1MAPTMPO
SCHEMBL1169735 0.71 HDAC8 (0.49) ADORA3ADORA2AADORA1MPOHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed