SCHEMBL20155113

SCHEMBL20155113

CCSNc1ccc(Nc2ccc(F)cc2F)c(-c2cn(C)c(=O)c3cn(Cc4ccccc4)nc23)c1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 16/20 0.48
THRB P10828 1/20 0.35
MEN1 O00255 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
BRD2 P25440 1/20 0.33
P2RX7 Q99572 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155652 0.90 BRD4 (0.48) BRD4BRD2
SCHEMBL20155659 0.85 BRD4 (0.46) BRD4THRBMEN1HTTKMT2A
SCHEMBL20155184 0.85 BRD4 (0.40) BRD4
SCHEMBL20155593 0.85 BRD4 (0.47) BRD4BRD2
SCHEMBL20155625 0.83 BRD4 (0.46) BRD4BRD2
SCHEMBL20155756 0.80 BRD4 (0.41) BRD4
SCHEMBL20155103 0.78 BRD4 (0.42) BRD4HTT
SCHEMBL20155168 0.77 BRD4 (0.40) BRD4
SCHEMBL20155116 0.76 BRD4 (0.45) BRD4
SCHEMBL20155467 0.75 BRD4 (0.50) BRD4BRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed